Discovery of GluN2A-Selective NMDA Receptor Positive Allosteric Modulators PAMs Tuning Deactivation Kinetics via StructureBased Design
Matthew Volgraf, Benjamin D. Sellers, Yu Jiang, Guosheng Wu, Cuong Q. Ly, Elisia Villemure, Richard M Pastor, Po-wai Yuen, Aijun Lu, Xifeng Luo, Mingcui Liu, Shun Zhang, Liang Sun, Yuhong Fu, Patrick J Lupardus, Heidi J A Wallweber, Bianca M. Liederer, Gauri Deshmukh, Emile Plise, Suzanne Tay, Paul Reynen, James Herrington, Amy Gustafson, Yichin Liu, Akim Dirksen, Matthias G A Dietz, Yanzhou Liu, Tzu-Ming Wang, Jesse Hanson, David Hackos, Kimberly Scearce-Levie, Jacob B. Schwarz
2016
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Journal of Medicinal Chemistry