Novel Alpha-7 Nicotinic Acetylcholine Receptor Agonists Containing a Urea Moiety: Identification and Characterization of the Potent, Selective, and Orally Efficacious Agonist 1-[6-(4-Fluorophenyl)pyridin-3-yl]-3-(4-piperidin-1-ylbutyl) Urea (SEN34625/WYE-103914)

Chiara Ghiron, Simon N. Haydar, Suzan Aschmies, Hendrick Bothmann, Cristiana Castaldo, Giuseppe Cocconcelli, Thomas A. Comery, Li Di, John Dunlop, Tim Lock, Angela Kramer, Dianne Kowal, Flora Jow, Steve Grauer, Boyd Harrison, Salvatore La Rosa, Laura Maccari, Karen L. Marquis, Iolanda Micco, Arianna Nencini, Joanna Quinn, Albert J. Robichaud, Renza Roncarati, Carla Scali, Georg C. Terstappen, Elisa Turlizzi, Michela Valacchi, Maurizio Varrone, Riccardo Zanaletti, Ugo Zanelli

2010
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Journal of Medicinal Chemistry

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